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  • 标题:Novel Cubosome System Resistant to Lipid Removal by Serum Albumin
  • 本地全文:下载
  • 作者:Makoto Uyama ; Tetsurou Handa ; Minoru Nakano
  • 期刊名称:Chemical and Pharmaceutical Bulletin
  • 印刷版ISSN:0009-2363
  • 电子版ISSN:1347-5223
  • 出版年度:2019
  • 卷号:67
  • 期号:10
  • 页码:1099-1103
  • DOI:10.1248/cpb.c19-00370
  • 出版社:The Pharmaceutical Society of Japan
  • 摘要:

    Cubosomes are lipidic nanoparticles containing bicontinuous cubic structures. Their unique architecture and potential as drug delivery vehicles have attracted researchers’ attention. However, cubosome systems that are more robust in the presence of plasma components are being sought after for applications in intravenous administration. In this study, we prepared cubosomes consisting of 1,2-dioleoyl- sn -glycero-3-hexylphosphocholine (hexyl-DOPC) and compared their interaction with bovine serum albumin (BSA), the most abundant protein in plasma, with that of conventional cubosome systems consisting of several bicontinuous cubic phase-forming lipids, including 1-monoolein (MO), 1- O -(5,9,13,17-tetramethyloctadecanoyl)erythritol (EROCO C22), or 1- O -(5,9,13,17-tetramethyloctadecyl)-β-D-xylopyranoside (β-XP). The average number of lipids bound to each BSA molecule was between 1.2–4.0 for MO, EROCO C22, and β-XP. On the other hand, hexyl-DOPC exhibited negligible binding to BSA. This result suggests that hexyl-DOPC, which was shown to resist removal from particles by BSA, can be used as a new lipid component of cubosomes, and has higher plasma stability than the other cubic phase-forming lipids.

  • 关键词:bicontinuous cubic phase;monoolein;hexylphosphocholine;serum albumin
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